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Development of Integrated Parent–Metabolite Pharmacokinetic Model With Apparent Presystemic Metabolism to Characterize the Disposition of Alverine
作者Ara Cho; Hyeon‐Cheol Jeong; MinJu Kim; Inkyung Cho; Hyeon‐Jeong Na; Kyong‐Cheol Ko; Yoon‐Jee Chae; Kyeong‐Ryoon Lee
作者单位1. Advanced Alternative Testing Team Korea Research Institute of Bioscience and Biotechnology Cheongju Republic of Korea; 2. Korea Preclinical Evaluation Center Korea Research Institute of Bioscience and Biotechnology Daejeon Republic of Korea; 3. Laboratory Animal Resource & Research Center Korea Research Institute of Bioscience and Biotechnology Cheongju Republic of Korea; 4. Department of Pharmacology, College of Medicine Konyang University Daejeon Republic of Korea; 5. Department of Bioengineering University of Science and Technology Daejeon Republic of Korea
Integrating CRRT as a Virtual Organ Into Physiologically Based Pharmacokinetic Modeling to Optimize Antimicrobial Dosing in Septic Patients
作者Yuanming Xing; Yijing Zhang; Chuqi Bai; Yulan Qiu; Chuhui Wang; Lei Chen; Taotao Wang; Jiaojiao Chen
作者单位1. Department of Cardiovascular Medicine The First Affiliated Hospital of Xi'an Jiaotong University Xi'an China; 2. Department of Pharmacy The First Affiliated Hospital of Xi'an Jiaotong University Xi'an China; 3. Department of Hemodialysis The First Affiliated Hospital of Xi'an Jiaotong University Xi'an China
Net Renal Drug Secretion Critically Requires Significant Contribution of Basal Uptake Transporters: Perspective From Mechanistic Kidney Model Simulation and Integration of Clinical and In Vitro Data
作者Toshiaki Tsuchitani; Masatoshi Tomi; Yuichi Sugiyama
作者单位1. Faculty of Pharmacy Keio University Tokyo Japan; 2. Genomembrane Co. Ltd Yokohama Kanagawa Japan; 3. iHuman Institute ShanghaiTech University Shanghai China
Model‐Based Tacrolimus Dosing Using the Population Pharmacokinetic Analysis Under the Nirmatrelvir/Ritonavir Therapy
作者Kotaro Itohara; Yoshiki Katada; Takahiro Hatayama; Toshiaki Igarashi; Jiro Ogura; Tomoki Fukushima; Shingo Yamazaki; Masato Homma; Takashi Niwa; Yoshiaki Kato; Nanae Yamamoto; Hideyuki Terazono; Hideo Shiohira; Tomohiro Terada; Ikuko Yano
作者单位1. Department of Pharmacy Kobe University Hospital Kobe Japan; 2. Department of Clinical Pharmacology and Therapeutics Kyoto University Hospital Kyoto Japan; 3. Department of Pharmacy Hirosaki University Hospital Hirosaki Japan; 4. Department of Pharmaceutical Sciences Tohoku University Hospital Sendai Japan; 5. Department of Pharmacy Yamagata University Hospital Yamagata Japan; 6. Department of Pharmacy University of Yamanashi Hospital Chuo Japan; 7. Division of Pharmacy Chiba University Hospital Chiba Japan; 8. Department of Pharmacy University of Tsukuba Hospital Tsukuba Japan; 9. Department of Pharmacy Gifu University Hospital Gifu Japan; 10. Department of Hospital Pharmacy Nagoya University Hospital Nagoya Japan; 11. Department of Pharmacy Kyushu University Hospital Fukuoka Japan; 12. Department of Pharmacy Kagoshima University Hospital Kagoshima Japan; 13. Department of Pharmacy University of the Ryukyus Hospital Ginowan Japan; 14. Laboratory of Clinical Pharmacy Showa Pharmaceutical University Machida Japan
Semi‐Mechanistic Modeling of S‐531011, a Humanized Anti‐ CCR8 Monoclonal Antibody, for Prediction of CCR8 Receptor Occupancy in Human Tumor Tissues
作者Daichi Yamaguchi; Wataru Nogami; Yudai Sonoda; Hitomi Morihara; Takayuki Katsube
作者单位1. Clinical Pharmacology and Pharmacokinetics Shionogi and Co., Ltd. Osaka Japan; 2. Laboratory for Drug Discovery and Development Shionogi and Co., Ltd. Osaka Japan
Pharmaceutical Industry Perspectives on Exposure‐Response Confounding in Large Molecule Therapeutics: Results From an IQ Consortium Survey
作者Engie Salama; Manisha Lamba; Sihem Ait‐Oudhia; Ellen Wang; Dorothee Semiond; Zhang Li; Tao Long; Satyendra Suryawanshi; Leticia Arrington; Wei Gao; Xiaowen Guan; Hugh Giovinazzo; Dale Miles; David C. Turner
作者单位1. Clinical Pharmacology & Pharmacometrics Xencor Pasadena California USA; 2. Pharmacometrics & Systems Pharmacology Pfizer Pearl River New York USA; 3. Quantitative Pharmacology and Pharmacometrics Merck & Co, Inc. Rahway New Jersey USA; 4. Translational Clinical Sciences, Internal Medicine Clinical Pharmacology Pfizer New York New York USA; 5. Sanofi R&D Cambridge Massachusetts USA; 6. Quantitative Clinical Pharmacology Daiichi Sankyo Basking Ridge New Jersey USA; 7. Takeda Development Center Americas, Inc. (TDCA) Cambridge Massachusetts USA; 8. Bristol Myers Squibb Princeton New Jersey USA; 9. Amgen Inc. Thousand Oaks California USA; 10. Moderna Therapeutics, Inc. Cambridge Massachusetts USA; 11. Regeneron Pharmaceuticals Tarrytown New York USA; 12. BeOne Medicines, Ltd San Carlos California USA; 13. Clinical Pharmacology Genentech South San Francisco California USA
Precision Dosing of Tacrolimus in Liver Transplantation: Integrating Donor‐Recipient CYP3A5 Pharmacogenomics and Drug Interactions
作者Virunya Komenkul; Prawat Chantharit; Piyawat Komolmit; Bunthoon Nonthasoot; Athaya Vorasittha; Anapat Sanpavat; Sirinporn Suksawatamnuay; Chandramouli Radhakrishnan; Thitima Wattanavijitkul
作者单位1. Department of Pharmacy Practice, Faculty of Pharmaceutical Sciences Chulalongkorn University Bangkok Thailand; 2. Department of Pharmaceutical Care, Faculty of Pharmacy Silpakorn University Nakorn Pathom Thailand; 3. Division of Infectious Diseases, Department of Medicine, Faculty of Medicine Ramathibodi Hospital, Mahidol University Bangkok Thailand; 4. Excellence Center in Liver Diseases King Chulalongkorn Memorial Hospital, Thai Red Cross Society Bangkok Thailand; 5. Department of Surgery, Faculty of Medicine Chulalongkorn University & King Chulalongkorn Memorial Hospital Bangkok Thailand; 6. Department of Pathology, Faculty of Medicine Chulalongkorn University and King Chulalongkorn Memorial Hospital Bangkok Thailand; 7. Certara Radnor Pennsylvania USA
Adjoint and Unrolled Automatic Differentiation for Laplace‐Approximated Likelihoods in Population PK and PK / PD Models
作者Guido H. Jajamovich; William Holmes; Chih‐Wei Lin; Khamir Mehta
作者单位1. Clinical Pharmacology Modeling and Simulation Amgen South San Francisco California USA; 2. Clinical Pharmacology Modeling and Simulation Amgen Thousand Oaks California USA
Transporter‐Drive Interstitial Tissue Exposure and Pharmacodynamic Response of Meropenem in Sepsis: A Mechanistic PBPK Modeling Study
作者Laura Ben Olivo; Jessica Luisa Silva de Lemos; Vinicius Jardim Rodrigues; Bibiana Verlindo de Araújo
作者单位1. Pharmaceutical Sciences Graduate Program Federal University of Rio Grande Do Sul Porto Alegre Brazil; 2. Biological Sciences Graduate Program: Pharmacology and Therapeutics Federal University of Rio Grande Do Sul Porto Alegre Brazil
Deciphering the Mechanisms of Statin–Ezetimibe Drug Combinations Using Boolean Logical Modeling and Transcriptomic Data
作者Rui‐Sheng Wang; Matteo Pedrelli; Osman Ahmed; Garagnani Paolo; Paolo Parini; Joseph Loscalzo
作者单位1. Department of Medicine Brigham and Women's Hospital Boston USA; 2. Cardio Metabolic Unit, Department of Medicine and Department of Laboratory Medicine Karolinska Institute Huddinge Sweden; 3. Medical Unit Endocrinology, Theme Inflammation and Ageing Karolinska University Hospital Stockholm Sweden; 4. Department of Biochemistry, College of Medicine and Health Sciences Arabian Gulf University Manama Kingdom of Bahrain; 5. Department of Experimental, Diagnostic and Specialty Medicine (DIMES) University of Bologna Bologna Italy
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