医学
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19 篇有效样本 · 按发表日期由新到旧排列
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An Ultra‐Fast UPLC‐MS/MS Method for Quantifying Ivosidenib: Application to Assessment of Metabolic Stability in Human Liver Microsomes
作者Mohamed W. Attwa; Ali S. Abdelhameed; Haitham AlRabiah; Adnan A. Kadi
作者单位1. Department of Pharmaceutical Chemistry College of Pharmacy Riyadh Saudi Arabia
New Chromene Derivatives as Promising VEGFR‐2 Inhibitors: Experimental Cytotoxicity and Comprehensive Computational Characterization
作者Hazem Elkady; Aisha A. Alsfouk; Eslam B. Elkaeed; Walid E. Elgammal; Hazem A. Mahdy; Ahmed Nofal; Ibrahim H. Eissa; Dalal Z. Husein; Fatma G. Amin; Ahmed M. Metwaly
作者单位1. Pharmaceutical Medicinal Chemistry & Drug Design Department, Faculty of Pharmacy (Boys) Al‐Azhar University Cairo Egypt; 2. Department of Pharmaceutical Sciences, College of Pharmacy Princess Nourah bint Abdulrahman University Riyadh Saudi Arabia; 3. Department of Pharmaceutical Sciences, College of Pharmacy AlMaarefa University Diriyah Riyadh Saudi Arabia; 4. Department of Chemistry Faculty of Science, Al‐Azhar University Nasr City Cairo Egypt; 5. Faculty of Pharmacy Al‐Azhar University Cairo Egypt; 6. Chemistry Department, Faculty of Science New Valley University El‐Kharja Egypt; 7. Physics Department, Faculty of Science Alexandria University Alexandria Egypt; 8. Pharmacognosy and Medicinal Plants Department, Faculty of Pharmacy (Boys) Al‐Azhar University Cairo Egypt
Metabolic Activation‐Dependent Anti‐Liver Cancer Activity and Organ‐Specific Toxicity of Retrorsine From Fanhuncao ( Jacobaea cannabifolia and J. litvinovii )
作者Zhijie He; Zhongyu Tan; Lunrong Zhang; Yue Yin; Yedeli Yerjiang; Bo Bi; Jingshan Bao
作者单位1. School of Pharmacy Changchun University of Chinese Medicine Changchun Jilin China; 2. College of Chinese Medicinal Materials Jilin Agricultural University Changchun Jilin China; 3. School of Clinical Medicine Changchun University of Chinese Medicine Changchun Jilin China; 4. School of Acupuncture and Tuina Changchun University of Chinese Medicine Changchun Jilin China
BRET‐Based Approaches for Ion Channels: Emerging Applications and Future Directions
作者Nadine Kock; Laura Heitzer; Joana Massa; Marvin Taterra; Marcel Bermúdez; Oliver Koch; Matthias Schiedel
作者单位1. Institute for Pharmaceutical and Medical Chemistry, Faculty of Chemistry and Pharmacy University of Münster Münster Germany; 2. GRK 2515, Chemical biology of ion channels (Chembion) Universität Münster Münster Germany
Discovery of Novel Ligands for the Treatment of Cryptococcus neoformans Infection
作者Teresa Rocha; Catarina Alves; Carla Lima; Lisa Sequeira; Fernanda Borges; Fernando Cagide; Sofia Benfeito
作者单位1. RISE‐Health, Departamento de Biomedicina Faculdade de Medicina da Universidade do Porto Porto Portugal; 2. Departamento de Química e Bioquímica Faculdade de Ciências da Universidade do Porto Porto Portugal
First UV‐Based Strategies Integrating Whiteness, Greenness, and Blueness Appraisals for Estimating Meloxicam and Tramadol Concurrently in Their Veterinary Mixture
作者Ahmed R. Mohamed; Eman Darweish; Sabry M. Attia; Tanveer Singh; Youstina M. Metias
作者单位1. Pharmaceutical Analytical Chemistry Department, Faculty of Pharmacy Egyptian Russian University Badr Cairo Egypt; 2. Department of Pharmacology and Toxicology, College of Pharmacy King Saud University Riyadh Saudi Arabia; 3. Department of Molecular and Integrative Physiology University of Illinois at Urbana‐Champaign Urbana Illinois USA; 4. Pharmaceutical Analytical Chemistry Department, Faculty of Pharmacy Zagazig University Zagazig Egypt
Recent Developments and Structure–Activity Relationships of BRAF Inhibitors for Cancer Drug Discovery
作者Xin‐Ke Guo; Kadalipura P. Rakesh; Sahana Raju; Kothanahally S. Sharath Kumar; Hua‐Li Qin
作者单位1. School of Chemistry, Chemical Engineering and Life Sciences Wuhan University of Technology Wuhan People's Republic of China; 2. Department of Physics, GSSS Institute of Engineering and Technology for Women, Metagalli, Mysuru Visvesvaraya Technological University, Belagavi Mysuru Karnataka India; 3. Department of Studies in Chemistry, Manasagangotri University of Mysore Mysuru India
Olikomycin A Disrupts Gram‐Positive Bacterial Membranes Through Calcium‐Dependent Binding to Phosphatidylglycerol
作者Luisa Munz; Olga Makshakova; Sara Marchi; Winfried Römer; Andreas Bechthold
作者单位1. Pharmaceutical Biology and Biotechnology Institute for Pharmaceutical Sciences University of Freiburg Freiburg Baden‐Württemberg Germany; 2. Synthetic Biology of Signaling Processes, Faculty of Biology University of Freiburg Freiburg Baden‐Württemberg Germany; 3. CIBSS – Centre for Integrative Biological Signaling Studies University of Freiburg Freiburg Baden‐Württemberg Germany
Targeting Human Protein Kinase CK2 by a Library of Indeno[1,2‐ b ]Indoles: Contribution of Thermal Shift Assay to Pre‐Screening and Co‐Crystallization to Post‐Screening
作者Matheus M. Guimarães; Christian Werner; Belen Leroy; Johana Charles; Jean Guillon; Noël Pinaud; Angélique Mularoni; Marc Jean‐Baptiste; Perrine Ximenes; Alexander Gast; Helge Prinz; Dagmar Aichele; Alan G. Gonçalves; Christelle Marminon; Zouhair Bouaziz; Joachim Jose; Jean‐Guy Delcros; Karsten Niefind; Marc Le Borgne
作者单位1. Gastroenterology and Technologies for Health Team, Centre de Recherche en Cancérologie de Lyon, Centre Léon Bérard, CNRS 5286, INSERM 1052 Université Claude Bernard Lyon 1, Univ. Lyon Lyon France; 2. Laboratory of Synthesis of Heterocycles and Glycoconjugates, Pharmaceutical Sciences Post‐Graduation Program Federal University of Paraná Curitiba Paraná Brazil; 3. Institute of Biochemistry, Department of Chemistry and Biochemistry University of Cologne Koln Germany; 4. INSERM, CNRS, ARNA, U1212, UMR 5320, UFR des Sciences Pharmaceutiques Univ. Bordeaux Bordeaux France; 5. ISM‐CNRS UMR 5255 Univ. Bordeaux Talence France; 6. Institute of Pharmaceutical and Medicinal Chemistry, PharmaCampus University of Münster Münster Germany; 7. Institut des Sciences Pharmaceutiques et Biologiques (ISPB), Faculté de Pharmacie Université Claude Bernard Lyon 1, Univ. Lyon Lyon France
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