Paper Review Records
All Paper Review Records
15 valid samples · Newest publication first
Review days = acceptance date − received date. PDF, DOI, and publisher-page sources are retained.
In silico and in vitro evaluation of new sulfonamide derivatives as VEGFR-2 inhibitors for cancer therapy
AuthorsAhmed Wheed Radhi; Hayder Ghanim Chfat; Zahraa Sabbar Omarn; Hayder Kadhim Abbas; Ali Jabbar Radhi; Ehab K. Obaid
Affiliations1. University of Kufa; 2. Jabir Ibn Hayyan University for Medical and Pharmaceutical Sciences; 3. Kerbala University; 4. University of Al-Kafeel; 5. ARCPMS, University of AlKafeel; 6. Al-Qasim Green University
Chalcone-indole hybrid scaffolds as promising anticancer drug candidates: a mini-review
AuthorsYafei Zhuang; Yanjing Cheng; Danchen Zhao; Jun Yu; Lianlian Chen
Affiliations1. Hubei University of Science and Technology
Design and development of 2,7-disubstituted 6-methoxyquinazolin-4 (3 H )-ones as potential anti-cancer agents possibly through downregulation of Wnt/β-catenin/TCF4 signaling pathway
AuthorsPrashant R. Murumkar; Kaushik Neogi; Premlal Meher; Rasana Yadav; Karan Joshi; Omkumar Prajapati; Priyanshu Sharma; Poonam Yadav; Devarajan Karunagaran; Prasanta Kumar Nayak; Mange Ram Yadav
Affiliations1. The Maharaja Sayajirao University of Baroda; 2. Indian Institute of Technology (Banaras Hindu University); 3. Indian Institute of Technology Madras; 4. Parul University
Advancing cancer drug discovery through the integration of machine learning and high-throughput screening
AuthorsKamil Herbetko; Katarzyna Herbetko; Magdalena Mikołajek; Laura Wojdyło; Karolina Klasen; Marek Kulbacki; Julita Kulbacka
Affiliations1. Wroclaw University of Science and Technology; 2. Wroclaw Medical University; 3. Wroclaw University of Environmental and Life Sciences; 4. Polish-Japanese Academy of Information Technology; 5. DIVE IN AI; 6. State Research Institute Centre for Innovative Medicine
Beyond the ATP-binding pocket: emerging strategies in kinase targeting from allosteric inhibition to targeted protein degradation
AuthorsMei Zhou; Linshan Li; Xiaojuan Tang; Yazhu Zhao; Wei Zhang
Affiliations1. Sichuan University; 2. Nursing Key Laboratory of Sichuan Province
Novel thioether and thioester-based derivatives as promising antibacterial agents with antioxidant potential: design, synthesis, and in silico studies
AuthorsAya H. Othman; Menna M. A. Abd El-Mageed; Faten Farouk; Ayman B. Farag; Safinaz E-S. Abbas
Affiliations1. Cairo University; 2. Ahram Canadian University; 3. University of Arizona
Rational drug design for Alzheimer’s disease: from approved therapies to next-generation clinical candidates and AI-guided innovation
AuthorsSana Saffour; Turgut Seckin Gul; Halise Inci Gul
Affiliations1. Atatürk University; 2. Trustlife Laboratories Drug Research & Development Center; 3. Ataturk University
Asymmetric benzazole derivatives as dual antibiofilm and anti-wall teichoic acid agents against Staphylococcus aureus
AuthorsMine Buga Aktekin; Zehra Oksuz; Mehmet Abdullah Alagoz; Bahar Uluca Han; Oztekin Algul
Affiliations1. Mersin University; 2. Tarsus University; 3. İnönü University; 4. Erzincan Binali Yıldırım University Yalnizbag Campus
Latest developments in small molecule inhibitors of cysteine protease B as antileishmanial drugs
AuthorsKarla Joane da Silva Menezes; Sonaly Lima Albino; João Vitor Vieira da Silva; Éric de Oliveira Rios; Rafaella Alves da Silva Barbosa; Juan D. Rodríguez-Macías; Edgar Alexander Marquez Brazon; Fátima Nogueira; Sofia Cortes; Ricardo Olimpio de Moura; Igor José dos Santos Nascimento
Affiliations1. Universidade Estadual da Paraíba (UEPB); 2. Universidade NOVA de Lisboa (UNL); 3. Universidade Estadual da Paraíba; 4. Centro Universitário Cesmac; 5. Exactas y Naturales, Universidad Libre; 6. Universidad del Norte; 7. Centro Universitário Estácio de Alagoas
Design, synthesis and dual anticancer and antibacterial evaluation of novel 1,3,4-oxadiazole-2-thiol derivatives targeting EGFR and DNA Gyrase B: integrated docking, DFT and ADMET studies
AuthorsIla M. Ram; Jay B. Maheta; Darshna K. Lakhnotra; Nargis H. Shaikh; Prince A. Dave; Parth Thakor; Shivani Lakhani; Anjali B. Thakkar; Yogesh O. Bhola
Affiliations1. Shri M.P. Pandya Science College, Shri Govind Guru University-Godhra; 2. Charotar University of Science and Technology; 3. Sardar Patel University
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