Paper Review Records
All Paper Review Records
25 valid samples · Newest publication first
Review days = acceptance date − received date. PDF, DOI, and publisher-page sources are retained.
131
days
Deconstruction of Aspartic Protease Inhibitors Enables Fragment‐Based Discovery of Plasmepsin V Inhibitors
Authors
Marija Skvorcova; Laura Ruduša; Diana Zelencova‐Gopejenko; Aigars Jirgensons; Raitis BobrovsShow moreShow less
Affiliations
1. Latvian Institute of Organic Synthesis Riga Latvia; 2. Molport Inc. Riga LatviaShow moreShow less
43
days
Novel Water‐Soluble, Heavy Atom‐Free Thioxanthene‐Fused Naphthalimide–Polyamine Phototheranostic Conjugates
Authors
Elisa Uliassi; Michele Rossi; Matteo Di Giosia; Amalia Conti; Matteo Calvaresi; Kerry J. Rhoden; Maria Laura BolognesiShow moreShow less
Affiliations
1. Department of Pharmacy and Biotechnology Alma Mater Studiorum ‐ University of Bologna Bologna Italy; 2. Department of Chemistry “Giacomo Ciamician” Alma Mater Studiorum ‐ University of Bologna Bologna Italy; 3. Preclinical & Translational Research in Oncology lab (PRO) IRCCS Azienda Ospedaliero ‐ Universitaria di Bologna Bologna Italy; 4. Medical Genetics Unit IRCCS Azienda Ospedaliero ‐ Universitaria di Bologna Bologna Italy; 5. Interdepartmental Center for Health Sciences & Technologies (HST), CIRI‐SDV Alma Mater Studiorum ‐ University of Bologna Bologna Italy; 6. Department of Medical and Surgical Sciences Alma Mater Studiorum ‐ University of Bologna Bologna ItalyShow moreShow less
158
days
Exploration of Nirmatrelvir Derivatives as Optimized SARS‐CoV‐2 Antivirals
Authors
Yugendar R. Alugubelli; Veerabhadra R. Vulupala; Kai S. Yang; Kaustav Khatua; Lauren R. Blankenship; Sathish Kumar; Demonta Coleman; Xuejiao Guo; Zhi Zachery Geng; Chia‐Chuan D. Cho; Banumathi Sankaran; Benjamin W. Neuman; Shiqing Xu; Wenshe Ray LiuShow moreShow less
Affiliations
1. Texas A&M Drug Discovery Center Department of Chemistry College of Arts and Sciences Texas A&M University College Station Texas USA; 2. Department of Biology College of Arts and Sciences Texas A&M University College Station Texas USA; 3. Molecular Biophysics and Integrated Bioimaging Berkeley Center for Structural Biology Laurence Berkeley National Laboratory Berkeley California USA; 4. Texas A&M Global Health Research Complex Texas A&M University College Station Texas USA; 5. Department of Molecular Pathogenesis and Immunology College of Medicine Bryan Texas USA; 6. Department of Pharmaceutical Sciences Irma Lerma Rangel College of Pharmacy Texas A&M University College Station Texas USA; 7. Institute of Biosciences and Technology Department of Translational Medical Sciences School of Medicine Texas A&M University Houston Texas USA; 8. Department of Biochemistry and Biophysics College of Agriculture and Life Sciences Texas A&M University College Station Texas USA; 9. Department of Cell Biology and Genetics College of Medicine Texas A&M University College Station Texas USAShow moreShow less
209
days
Design and Synthesis of Morroniside Derivatives Targeting H 2 O 2 ‐Induced Oxidative Stress: Antioxidant‐Triggered Neuroprotective Effect
Authors
Mingtao Wang; Haiyi Gao; Yuxiang Song; Baohong Sun; Yian Zhao; Peiliang Dong; Hua HanShow moreShow less
Affiliations
1. College of Medicine Heilongjiang University of Chinese Medicine Harbin China; 2. Institute of Traditional Chinese Medicine Heilongjiang University of Chinese Medicine Harbin ChinaShow moreShow less
133
days
Rational Design of Multifunctional Tacrine Derivatives as Candidates for the Treatment of Alzheimer and Parkinson Diseases
Authors
Eugenia Dzib; Luis Felipe Hernández‐Ayala; Silvana Silva‐Aguirre; Annia GalanoShow moreShow less
Affiliations
1. Departamento de Química División de Ciencias Básicas e Ingeniería Universidad Autónoma Metropolitana, Unidad Iztapalapa Ciudad de México México; 2. Departamento de Física Aplicada Centro de Investigación y de Estudios Avanzados, Unidad Mérida Mérida Yucatán MéxicoShow moreShow less
72
days
Hydroamination of Dehydroalanine With Deuterium Incorporation to Access Unnatural 2‐ and 4‐Pyridonyl α‐Amino Acids: Evaluation of Their Antibacterial, Antifungal, and Immunomodulatory Activities
Authors
Sowmya B. Udayakumar; Prakash Kumar; Karnati Sai Pranathi; Anjali Prajapati; Sunil Misra; Srinivasa Reddy Bonam; Kiranmai NayaniShow moreShow less
Affiliations
1. Department of Organic Synthesis and Process Chemistry CSIR‐Indian Institute of Chemical Technology Hyderabad India; 2. Academy of Scientific and Innovative Research (AcSIR) Ghaziabad India; 3. Department of Applied Biology CSIR‐Indian Institute of Chemical Technology Hyderabad India; 4. Vaccine Immunology Laboratory Department of Applied Biology CSIR‐Indian Institute of Chemical Technology Hyderabad IndiaShow moreShow less
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