医学
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Imidazo[1,2-a]pyridine-based HDAC6 inhibitor a17 for the treatment of Alzheimer's disease
作者Zhe Han; Wenmin Liu; Wenling Fu; Keren Wang; Zhenghuai Tan; Dongwei Zhang; Feifei Yang; Wu Dong; Zhipei Sang
作者单位College of Animal Science and Technology, Inner Mongolia Minzu University, Tongliao, 028000, China; College of Chemistry and Pharmaceutical Engineering, Nanyang Normal University, Nanyang, 473061, China; Key Laboratory of Tropical Biological Resources of Ministry of Education and and Hainan Engineering Research Center for Drug Screening and Evaluation, School of Pharmaceutical Sciences, Hainan University, Haikou, 570228, China; Institute of Traditional Chinese Medicine Pharmacology and Toxicology, Sichuan Academy of Chinese Medicine Sciences, Chengdu, 610041, China; Affiliated Hospital of Inner Mongolian Minzu University, Tongliao, Inner Mongolia, 02800, China; Pharmacy College, Henan University of Chinese Medicine, Zhengzhou, 450046, China
A novel cyclic-peptide antagonist of TIM-3 for cancer immunotherapy by reinvigorating exhausted T-cell activity
作者Ying Huang; Jiale Li; Yingzhou Qin; Bo Qie; Qianqian Wang; Cuijuan Liu; Yimin Zhu
作者单位School of Nano-Tech and Nano-Bionics, University of Science and Technology of China, Hefei, 230026, China; Division of Nano Biomedicine, Suzhou Institute of Nano-Tech and Nano-Bionics, Chinese Academy of Sciences, Suzhou, 215123, China; Nano-Bio-Chem Centre, Suzhou Institute of Nano-tech and Nano-bionics, Chinese Academy of Sciences, Suzhou, 215123, China
Class-specific and cumulative effects of psychotropic medication on sleep architecture: a polysomnographic retrospective study
作者Daniel Alfaiate; Patrícia Silva; Patrícia Guerra; Nuno Pinto; Alexandre Pereira
作者单位Polytechnic University of Castelo Branco, Castelo Branco, Portugal; Médio Tejo Local Health Unit, Torres Novas, Portugal; Department of Pediatric Neurology, University Children's Hospital Zurich, Zurich, Switzerland; Faculty of Health Sciences, University of Beira Interior, Covilhã, Portugal; RISE-Health-UBI, University of Beira Interior, Covilhã, 6201-506, Portugal
The role and mechanism of rosiglitazone in endothelial-to-mesenchymal transition in pulmonary hypertension
作者Aoxue Yuan; Yaqian Bai; Yuanhang Jiang; Shengnan Si; Pengwei Wang; Fanrong Zhao; Yujing Chen; Tiantian Zhu
作者单位School of Pharmacy, Henan Medical University, Xinxiang, 453003, China; School of Pharmaceutical Sciences, Jilin University, Changchun, 130021, China; Department of Clinical Pharmacy, The First Affiliated Hospital of Henan Medical University, Xinxiang, 453100, China; Henan International Joint Laboratory of Cardiovascular Remodeling and Drug Intervention, Xinxiang, 453003, China
Zonisamide improves cognitive impairment and psychiatric symptoms related with SAPAP3 in mouse models of Alzheimer's disease
作者Fangtai Yi; Jianfeng Ma; Ruiyue Zhao; Qiuyu Xie; Sitong Lu; Kailong Zhang; Zuodong Zhong; Huijuan OuYang; Yuan Qin; Mingheng Xu; Qin Xue; Xinlu Wang; Wei Wei; Yinghua Liu
作者单位Department of Pharmacology, Guangzhou Municipal and Guangdong Provincial Key Laboratory of Molecular Target & Clinical Pharmacology, Guangzhou Medical University, Guangzhou, Guangdong, 511436, China; Key Laboratory of State Administration of Traditional Chinese Medicine of China, Department of Pathophysiology, School of Medicine, Institute of Brain Research, Jinan University, Guangzhou, Guangdong, 511443, China; Department of Nuclear Medicine, The First Affiliated Hospital of Guangzhou Medical University, Guangzhou, Guangdong, 510120, China
Preclinical characterization of the efficacy and safety of histamine H3 receptor antagonist, LINS01022, as a novel analgesic for chronic neuropathic pain treatment
作者Magdalena Maciuszek; Magdalena Białoń; Mateusz Królewski; Karolina Noworyta; Nathalia A. Fiocchi; Flavia B. Lopes; Katarzyna Starowicz; Wesley L. Gouveia; Lidia M. Lima; João Paulo S. Fernandes; Katarzyna Popiolek-Barczyk
作者单位Department of Neurochemistry, Maj Institute of Pharmacology, Polish Academy of Sciences, Krakow, Poland; Department of Pharmaceutical Sciences, Federal University of São Paulo, Diadema, SP, Brazil; Department of Medicine, Federal University of São Paulo, São Paulo, SP, Brazil; Laboratório de Avaliação e Síntese de Substâncias Bioativas (LASSBio®), Institute of Biomedical Sciences, Federal University of Rio de Janeiro, Rio de Janeiro, RJ, Brazil
Gallic acid, renal redox balance and NRF2-Related transcript-level modulation in a rat model of contrast-associated acute kidney injury
作者Nurhan Akyürek Bayhan; Demet Gündüz; Nasıf Fatih Karakuyu; İlter İlhan; Muhammet Yusuf Tepebaşi; Orhan Berk İmeci̇; Emine Sarman; Mehtap Savran
作者单位Department of Radiology, Faculty of Medicine, Suleyman Demirel University, Isparta, Turkey; Department of Radiology, Faculty of Medicine, Akdeniz University, Antalya, Turkey; Department of Pharmacology, Faculty of Pharmacy, Suleyman Demirel University, Isparta, Turkey; Department of Biochemistry, Faculty of Medicine, Suleyman Demirel University, Isparta, Turkey; Department of Medical Genetics, Faculty of Medicine, Suleyman Demirel University, Isparta, Turkey; Department of Pharmacology, Faculty of Medicine, Suleyman Demirel University, Isparta, Turkey; Department of Histology and Embryology, Faculty of Medicine, Afyonkarahisar Health Sciences University, Afyonkarahisar, Turkey
Intergenerational consequences of valproic acid exposure: Dose- and sex-specific effects in Drosophilamelanogaster
作者Silvana Hof-Michel; Belén Olga Ferrando Hernandez; Andreas Vilcinskas; Anika E. Wagner
作者单位Institute of Nutritional Science, Justus Liebig University, Giessen, Germany; Department of Food Technology, Food Sciences and Nutrition, Campus of International Excellence, “Campus Mare Nostrum”, University of Murcia, Murcia, Spain; Branch Bioresources, Fraunhofer Institute for Molecular Biology and Applied Ecology IME, Giessen, Germany; Institute for Insect Biotechnology, Justus Liebig University, Giessen, Germany; Center for Sustainable Food Systems, Justus Liebig University, Giessen, Germany
Sodium butyrate alleviates neuronal ferroptosis after gas explosion-induced traumatic brain injury via regulation of JNK/P38 MAPK signaling pathway
作者Xinwen Dong; Zheng Luo; Cuiying Li; Jie Gao; Yue Ma; Xiaoran Ma; Jiahang Yang; Sanqiao Yao; Weidong Wu; Yichun Bai; Qunwei Zhang; Wenjie Ren
作者单位Department of Environmental and Occupational Health, School of Public Health, Henan Medical University, Xinxiang, Henan, 453003, China; Department of Clinical Medicine, Junji College, Henan Medical University, Xinxiang, Henan, 453003, China; Department of Environmental and Occupational Health Sciences, School of Public Health and Information Sciences, University of Louisville, Louisville, KY, United States; Institutes of Health Central Plains, Henan Medical University, 601 Jinsui Street, Xinxiang, Henan, 453003, China
Binding capacity of Intravenous immunoglobulin G to BK polyomavirus determines its anti-BK polyomavirus activity in infected cultures
作者Noriaki Sato; Atsuko Shiraki; Masaya Takemoto; Yoshinori Takemura; Kaoru Sakai; Shota Fukae; Mitsuru Saito; Kazunari Tanabe; Seiya Imoto; Motoko Yanagita; Kimiyasu Shiraki
作者单位Division of Health Medical Intelligence, Human Genome Center, The Institute of Medical Science, The University of Tokyo, Tokyo, Japan; Department of Nephrology, Graduate School of Medicine, Kyoto University, Kyoto, Japan; Department of Anesthesiology, Graduate School of Medicine, Kyoto University, Kyoto, Japan; Department of Microbiology, Faculty of Pharmaceutical Sciences, Hokuriku University, Kanazawa, Japan; Department of Anesthesiology, Toyama University Hospital, Toyama, Japan; Department of Urology, Graduate School of Medicine, Osaka University, Osaka, Japan; Department of Urology, Akita University Hospital, Akita, Japan; Kidney Transplant Center/Robot Surgery Center, Shonan Kamakura General Hospital, Kanagawa, Japan; Faculty of Nursing, Senri Kinran University, Suita, Osaka, Japan; Hokuriku Health Service Association, Toyama, Japan
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