医学
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The top-down Finite Time Pharmacokinetic (FTPK) models vis-a-vis the bottom-up PBPK models in early drug development
作者Panos Macheras; Nikos Alimpertis; Athanasios A. Tsekouras
作者单位Faculty of Pharmacy, Laboratory of Biopharmaceutics Pharmacokinetics, National and Kapodistrian University of Athens, Athens, Greece; Finite Absorption Time (F.A.T.) Laboratories, National and Kapodistrian University of Athens, Athens, Greece; Department of Chemistry, Laboratory of Physical Chemistry, National and Kapodistrian University of Athens, Athens, Greece
Lipid nanoparticles for ursodeoxycholic acid delivery: A strategy for topical applications
作者Giada Mondanelli; Vincenzo Falcone; Roberto Sauri; Bruno Cerra; Marco Gargaro; Maurizio Ricci; Aurélie Schoubben; Antimo Gioiello
作者单位Department of Pharmaceutical Sciences, University of Perugia, Perugia, Italy
M4 drug discovery: Human drug predictions from integrated preclinical insights exemplified with a GLP-1R agonist
作者Oscar Silfvergren; Sophie Rigal; Katharina Schimek; Christian Simonsson; Kajsa P Kanebratt; Felix Forschler; Burcak Yesildag; Uwe Marx; Liisa Vilén; Peter Gennemark; Gunnar Cedersund
作者单位Department of Biomedical Engineering, Linköping University, Linköping, Sweden; SUND sound medical decisions, Linköping, Sweden; TissUse GmbH, Berlin, Germany; Institute of Biotechnology, Technische Universität Berlin, Berlin, Germany; Drug Metabolism and Pharmacokinetics, Research and Early Development, Cardiovascular, Renal and Metabolism (CVRM), BioPharmaceuticals R&D, AstraZeneca, Gothenburg, Sweden; InSphero AG, Schlieren, Switzerland; Bioscience Technology Research and Early Development, Cardiovascular, Renal and Metabolism (CVRM), BioPharmaceuticals R&D, AstraZeneca, Gothenburg, Sweden; Center for Medical Image Science and Visualization (CMIV), Linköping University, Linköping, Sweden; School of Medical Sciences and Inflammatory Response and Infection Susceptibility Centre (iRiSC), Faculty of Medicine and Health, Örebro University, Örebro, Sweden
Evaluation of Citicoline-loaded Lutrol 127/Carbopol/Hyaluronic acid-based gels for brain delivery by intranasal administration
作者Anna Patrizia de Nichilo; Francesca Uberti; Adriana Trapani; Stefano Castellani; Giorgia Iaconisi; Giorgia Franzino; Cinzia Di Franco; Lorenzo Guerra; Rosanna Mallamaci; Rosa Angela Cardone; Carmelo Ventra; Domenico Larobina; Loredana Capobianco; Simone Mulè; Elvira De Giglio
作者单位Department of Pharmacy-Drug Sciences, University of Bari “Aldo Moro”, via E. Orabona, Bari, 4-70125, Italy; Department for Sustainable Development and Ecological Transition, University of Piemonte Orientale (UPO), Piazza Sant’Eusebio 5, Vercelli, 13100, Italy; Department of Precision and Regenerative Medicine and Ionian Area (DiMePRe-J), University of Bari “Aldo Moro”, Bari, 70125, Italy; Department of Biological and Environmental Science and Technology, University of Salento, Via Lecce—Monteroni, Lecce, 73100, Italy; Consiglio Nazionale delle Ricerche Istituto per i Polimeri, Compositi e Biomateriali P. le Enrico Fermi, Naples, 1 80055, Italy; CNR-IFN Bari, Bari Via Amendola 173, 70126 Bari, Italy; Department of Biosciences, Biotechnologies and Environment, University of Bari “Aldo Moro”, Bari, 70125, Italy; Esseti Farmaceutici, Via Cavalli di Bronzo, 39-46, San Giorgio a Cremano, Naples, 80046, Italy .; Department of Chemistry, University of Bari “Aldo Moro”, Bari, 70125, Italy
FcBP-HFQ lipid-mediated trastuzumab modification of mRNA-loaded lipid nanoparticles enhances delivery to HER2-expressing cancer cells
作者Makoto Matsumoto; Riku Takayama; Chiemi Matsuguchi; Haruki Shimada; Tatsunori Izumi; Naoya Kato; Ayaka Matsuo-Tani; Hikaru Nakamura; Takeshi Hiu; Takayuki Matsuo; Hidefumi Mukai; Shigeru Kawakami
作者单位Graduate School of Biomedical Sciences, Nagasaki University, Nagasaki, Japan; Department of Neurosurgery, Graduate School of Biomedical Sciences, Nagasaki University, Japan
Differential myocardial responses to indobufen and aspirin across clinical and experimental models of myocardial infarction
作者Bryan Richard Sasmita; Bi Huang; Jiejie Yang; Suxin Luo; Yongzheng Guo
作者单位Department of Cardiology, Cardiovascular Research Center, The First Affiliated Hospital of Chongqing Medical University, Chongqing, 400016, China; Key Laboratory of Circulatory System Stress and Disease of Chongqing Municipal Education Commission, Chongqing Medical University, Chongqing, 400016, China
Discovery of a Potent and Selective KRAS G12D Degrader based on PROTAC Degradation
作者Lili Jiang; Wenyan Yang; Yanqing Liu; Gangjian Li; Xiaomin Luo; Yubo Zhou; Jiangjiang Qin; Youlu Pan; Wenhai Huang
作者单位Center of Safety Evaluation and Research, Key Laboratory of Drug Safety Evaluation and Research of Zhejiang Province, Hangzhou Medical College, Hangzhou, Zhejiang, 310053, China.; School of Pharmaceutical Sciences, Hangzhou Medical College, Hangzhou 310000, China.; Zhuji People's Hospital of Zhejiang Province, Zhuji 311800, China.; Center for Innovative Drug Research, Hangzhou Institute of Medicine (HIM), Chinese Academy of Sciences, Hangzhou, Zhejiang, China.; Zhongshan Institute for Drug Discovery, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Zhongshan, Guangdong 528400, China.; University of Chinese Academy of Sciences, Beijing, China.; School of Pharmacy, Faculty of Medicine, Macau University of Science and Technology, Macau 999078(or Macau SAR), China.
Synthesis and biological evaluation of 68Ga-DOTA-PLE: a Plectin-1-targeted radiotracer for PET/MR imaging of pancreatic cancer
作者Zhi-Qiang Yu; Hongrui Shu; Yujie Wang; Shun Li; Zhen-Peng Yu; Weijia Zhao; Xue-Feng Zhao; Hong Zhu; Yi Du; Pai Peng; Hongwei Si; Peng-Fei Dai
作者单位Department of Nuclear Medicine, The First Affiliated Hospital of Anhui Medical University, Hefei, Anhui, 230022, China; School of Life Sciences, Anhui Medical University, Hefei, Anhui, 230032, China; Department of Dermatology, The First Affiliated Hospital of Anhui Medical University, Hefei, Anhui, 230022, China; Anhui province key laboratory of tumor immune microenvironment and immunotherapy, The First Affiliated Hospital of Anhui Medical University, Hefei, Anhui, 230022, China; Department of Respiratory and Critical Care Medicine, The First Affiliated Hospital of Anhui Medical University, Hefei, Anhui, 230022, China
GW0742 prevents neointima formation by upregulating FABP3 expression
作者Xuesheng Wang; Jingjie Chen; Bo Huo; Xingliang Wu; Wenxin Lin; Ding-Sheng Jiang; Yu-Song Zhang; Xin Feng; Fu-Han Gong
作者单位Department of Cardiology, Tongren People's Hospital, Tongren, Guizhou, China; Division of Cardiovascular Surgery, Tongji Hospital, Tongji Medical College, Huazhong University of Science and Technology, Wuhan, Hubei, China; Key Laboratory of Organ Transplantation, Ministry of Education, Chinese Academy of Medical Sciences; NHC Key Laboratory of Organ Transplantation, Wuhan, Hubei, China
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