医学
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Development of Netrin-1-targeted peptide probes derived from the Netrin-1/DCC complex for noninvasive imaging of tumors
作者Shu Li; Shuang Wang; Xue Zhu; Zhihong Huang; Yang Jiao; Jiayuan Du; Jie Tang; Zhenfeng Liu; Ke Wang; Jing Fang
作者单位National Health Commission Key Laboratory of Nuclear Medicine, Jiangsu Key Laboratory of Molecular Nuclear Medicine, Jiangsu Institute of Nuclear Medicine, Wuxi, Jiangsu 214063, China; Department of Radiopharmaceuticals, School of Pharmacy, Nanjing Medical University, Nanjing 211166, China; Department of Nuclear Medicine, The First Affiliated Hospital, Zhejiang University School of Medicine, Hangzhou 310003, Zhejiang Province, China
Curculigoside suppresses glioblastoma progression through the EGFR/MMP2 axis: evidence from network pharmacology and experimental validation
作者Jiawen Han; Zhanchuan Ma; Shan Lin; Wei Wu
作者单位Central Laboratory, The First Hospital of Jilin University, Changchun, Jilin 130031, China; Key Laboratory of Organ Regeneration and Transplantation Ministry of Education, Changchun, Jilin 130021, China; Department of Respiratory Medicine, The First Hospital of Jilin University, Changchun, Jilin 130031, China; Department of Neurovascular Surgery, The First Hospital of Jilin University, Changchun, Jilin 130021, China
Discovery of Emodin as a novel competitive KPC-2 inhibitor through virtual screening: Synergistic efficacy with Meropenem against Carbapenem-resistant Klebsiella pneumoniae infection
作者Yan Wang; Jiamin Geng; Bingyan Li; Xuming Deng; Jiaxi Wang; Na Guo
作者单位College of Food Science and Engineering, Jilin University, Changchun 130062, China; State Key Laboratory for Diagnosis and Treatment of Severe Zoonotic Infectious Diseases, Key Laboratory for Zoonosis Research of the Ministry of Education, Institute of Zoonosis, and College of Veterinary Medicine, Jilin University, Changchun 130062, China
A honokiol-derived cationic amphiphilic compound combats methicillin-resistant Staphylococcus aureus by disrupting membrane phospholipid homeostasis
作者Muchen Zhang; Yan Wang; Jing Pan; Shengnan Xu; Shangshang Qin; Yanjiang Shao; Yong Guo
作者单位School of Pharmaceutical Sciences, Zhengzhou University, Zhengzhou 450001, Henan, China; School of Computer Science and Artificial Intelligence, Zhengzhou University, Zhengzhou, Henan 450001, China; Hunan Province Cooperative Innovation Center for Molecular Target New Drug Study, School of Pharmaceutical Science, Hengyang Medical School, University of South China, Hengyang 421001, China
Synthesis, multi-target enzyme inhibition, and in silico evaluation of phthalimide derivatives with relevance to tuberculosis-associated pathophysiology
作者Aneela Khushal; Sara Khan; Umar Farooq; Muhammad Naseem Khan; Misbah Hafeez; Rizwana Sarwar
作者单位Department of Chemistry, COMSATS University Islamabad, Abbottabad Campus, KPK, Pakistan; Department of Chemistry, Pennsylvania State University, University Park 16802, PA, USA
Dual-response mitochondria-targeted fluorescent probe for Hypochlorous acid and viscosity: Applications in liver injury diagnosis and environmental monitoring
作者Peng Hou; Qi Zhang; Junqiang Liu; Haoqing Ren; Pengfei Qi; Huiling Hou; Song Chen
作者单位College of Pharmacy, Qiqihar Medical University, Qiqihar 161006 , PR China; Achievement Transformation Center, Qiqihar Medical University, Qiqihar 161006, PR China
Structure-based optimization, in vitro profiling, and ADMET prediction of Celastrol derivatives as potent prolyl endopeptidase inhibitors
作者Tian-Ge Wang; Jing Zhang; Chang Dai; Wei-Ran Huang; Xiao-Lei Zhu; Kun-Jie Bian; Xian-Ting Jiao; Xing-Kai Qian; Li-Wei Zou
作者单位Department of Pediatric infectious, Xinhua Hospital Affiliated to Shanghai Jiao Tong University School of Medicine, Shanghai, China; Translational Medicine Research Center, Guizhou Medical University, 550025 Guiyang, Guizhou, China; Institute of Interdisciplinary Integrative Medicine Research, Shanghai University of Traditional Chinese Medicine, Shanghai 201203, China; Anshan Teachers Training Institute, Anshan 114000, China
A light-gated “membrane-to-mitochondria” sequentially targeted AIE photosensitizer for potentiated photodynamic therapy and imaging of breast cancer
作者Tonghui Huang; Fangzhu Huang; Nian Shi; Xing Wang; Hangying Ning; Li Lu; Cuiping Han
作者单位Department of Radiology, Affiliated Hospital of Xuzhou Medical University, Xuzhou 221004, China; School of Medical Imaging, Xuzhou Medical University, Xuzhou 221004, China; School of Pharmacy, Xuzhou Medical University, Xuzhou 221004, China
Fragment-based discovery of novel Baicalein derivatives as triple-target 3CLpro/PLpro/RdRp inhibitors against SARS-CoV-2
作者Di Han; Hongkun Yang; Yifan Wang; Fengxiang Liu; Wenfeng Lu; Baoyi Fan; Yuxiao Chang; Meiting Wang; Jiarui Lu; Taigang Liu; Shaoli Cui; Junqiang Zhao; Qinghe Gao; Jingqiang Cui; Yongtao Xu
作者单位School of Medical Engineering, Henan Medical University, Xinxiang, Henan 453003, China; Henan International Joint Laboratory of Neural Information Analysis and Drug Intelligent Design, Xinxiang, Henan 453003, China; Xinxiang Key Laboratory of Biomedical Information Research, Xinxiang, Henan 453003, China; School of Forensic, Henan Medical University, Xinxiang, Henan 453003, China; School of Medical Imaging, Henan Medical University, Xinxiang, Henan 453003, China; School of Pharmacy, Henan Medical University, Xinxiang, Henan, 453003, China; Henan Tuoren Medical Device Co., Ltd., Tuoren Industrial Zone, No. 1 Yangze Road, Changyuan County, 453400 Xinxiang, Henan, China
Design and synthesis of tenofovir monophenyl ester phosphonoamidate prodrugs with improved anti-hepatitis B virus activity and intrahepatic tenofovir enrichment
作者Xiaolei Wang; Sai Li; Ning Xu; Yundong Sun; Delong Liu; Jun Yu; Songgu Wu; Junbo Gong
作者单位School of Chemical Engineering and Technology, State Key Laboratory of Chemical Engineering, Tianjin University, Tianjin 300072, China; Jiangsu Hansoh Pharmaceutical Group Co., Ltd, Jiangsu 222047, China
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