医学
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20 篇有效样本 · 按发表日期由新到旧排列
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Targeting CDK‐2 With Novel Indole‐Pyrazole Hybrids: Discovery of Potent Anticancer Agents Supported by Mechanistic and In Silico Studies
作者Wagdy M. Eldehna; Zainab M. Elsayed; Mohamed R. Elnagar; Yasser M. Omar; Maha‐Hamadien Abdulla; Abdulrahman M. Saleh; Abdelrahman R. Shalabi; Diaaeldin M. Elimam; Suliman Alshamari; Mohamed Fares; Haytham O. Tawfik
作者单位1. Department of Pharmaceutical Chemistry, Faculty of Pharmacy Kafrelsheikh University Kafrelsheikh Egypt; 2. Scientific Research and Innovation Support Unit, Faculty of Pharmacy Kafrelsheikh University Kafrelsheikh Egypt; 3. Department of Pharmacology and Toxicology, Faculty of Pharmacy Al‐Azhar University Cairo Egypt; 4. Department of Pharmacology, College of Pharmacy The Islamic University Najaf Iraq; 5. Institute of Cancer Therapeutics University of Bradford Bradford UK; 6. Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy Assiut University Assiut Egypt; 7. Colorectal Research Chair, Department of Surgery, College of Medicine King Saud University Riyadh Saudi Arabia; 8. Postgraduate Program in Pharmaceutical Chemistry, Faculty of Pharmacy Cairo University, Cairo University Cairo Egypt; 9. Pharmaceutical Chemistry Department, Faculty of Pharmacy Sinai University North Sinai Egypt; 10. Department of Pharmacognosy, Faculty of Pharmacy Kafrelsheikh University Kafrelsheikh Egypt; 11. Sydney Pharmacy School The University of Sydney Sydney New South Wales Australia; 12. Department of Pharmaceutical Chemistry, Faculty of Pharmacy Tanta University Tanta Egypt; 13. Department of Pharmaceutical Chemistry, Faculty of Pharmacy Alsalam University Tanta Egypt
Alternative Splicing in Cyclin‐Dependent Kinase 4/6 Inhibitor Resistance in Estrogen Receptor‐Positive Breast Cancer
作者Yuqiu Cui; Jia Xie; Jiale Cai; Yue Si; Hairong Huang; Shiyi Yu; Haibo Sun
作者单位1. School of Medicine (Institute of Translational Medicine) Yangzhou University Yangzhou China; 2. Jiangsu Key Laboratory of Noncoding RNA Fundamental and Clinical Translational Research Yangzhou China
Applications of Bioinorganic Nano‐Based Delivery Systems—Diagnostics and Therapeutics
作者Frank Ssengooba; Jubilee Andrew; Donald Fernandes
作者单位1. Department of Pharmacy Practice, School of Pharmacy Sefako Makgatho Health Sciences University Pretoria South Africa; 2. Department of Pharmaceutical Sciences, School of Pharmacy Sefako Makgatho Health Sciences University Pretoria South Africa; 3. Department of Chemistry and Biology Toronto Metropolitan University Toronto Ontario Canada
GRP78 Drives NSCLC Stemness and EMT via a SIX1/β‐Catenin Signaling Axis
作者Guoping Tong; Huanyu Qi
作者单位1. Department of Respiratory and Tumor Internal Medicine, Chinese Academy of Medical Sciences Cancer Hospital Shanxi Hospital Shanxi Cancer Hospital Taiyuan City Shanxi Province China; 2. Department of Bone and Soft Tissue Tumor Oncology, Chinese Academy of Medical Sciences Cancer Hospital Shanxi Hospital Shanxi Cancer Hospital Taiyuan City Shanxi Province China
Two Novel 1,4‐Naphthoquinone Derivatives as Potent Agents Against Multidrug‐Resistant Staphylococcus aureus and Pathogenic Gram‐Positive Bacteria
作者HyunChan Song; Haena Lee; Ji‐Hyun Yoon; Hyunkyung Choi; Hakwon Kim; Ki‐Young Kim
作者单位1. Graduate School of Biotechnology Kyung Hee University Yongin Republic of Korea; 2. Department of Applied Chemistry, Global Center for Pharmaceutical Ingredient Materials Kyung Hee University Yongin Republic of Korea
Discovery of a Potent and Selective MAO‐B Inhibitor From a Donepezil‐Linked Chalcone Library With Promising Antiparkinsonian Activity
作者Azize Kirac‐Aydin; Bishnu Prasad Pandey; Satyajit Mohanty; Rupsa Mondal; Abanish Biswas; Ashok Kumar Pattnaik; Subodh Mondal; Vinay N. Basavanakatti; Nilüfer Bayrak; Venkatesan Jayaprakash; Hoon Kim; Amaç Fatih TuYuN
作者单位1. Department of Chemistry, Faculty of Science Istanbul University Istanbul Türkiye; 2. Institute of Graduate Studies in Science Istanbul University Istanbul Türkiye; 3. Department of Pharmacy College of Pharmacy, Sunchon National University Suncheon Republic of Korea; 4. Department of Chemical Science and Engineering Kathmandu University Kavre Nepal; 5. Department of Pharmaceutical Sciences and Technology Birla Institute of Technology Ranchi India; 6. Bioanalysis, Eurofins Advinus Biopharma Services India Pvt. Ltd Bengaluru India; 7. Adgyl Lifesciences Private Limited Bengaluru India
Ameliorative Effects of a Naphthoquinone Derivative With β‐Amyloid Aggregation Inhibitory Activity on Cognitive Impairment and Metabolite Analysis of the Blood and Brains of Mice
作者Jong Min Oh; Won Kyeong Jeong; Hyun Ju Son; Seo Young Kim; Tae Woo Oh; Moongi Ji; Ji Woo Nam; Minyeong Baek; Jeong‐Ho Park; Woong‐Hee Shin; Hee Jung Kim; Byeongchan Choi; Man‐Jeong Paik; Hoon Kim
作者单位1. Department of Pharmacy, College of Pharmacy Sunchon National University Suncheon Republic of Korea; 2. Herbal Medicine Resources Research Center Korea Institute of Oriental Medicine Naju Republic of Korea; 3. Korean Medicine (KM) Application Center, Korea Institute of Oriental Medicine (KIOM) Daegu Republic of Korea; 4. University of Science and Technology (UST), Korean Convergence Medicine Major KIOM Daejeon Republic of Korea; 5. Department of Chemical & Biological Engineering Hanbat National University Daejeon Republic of Korea; 6. Department of Biomedical Informatics, College of Medicine Korea University Seoul Republic of Korea
Discovery of Novel PCSK9‐LDLR PPI Inhibitors by a Structural Modification Approach
作者Huan Zhu; Zhiqin Zhang; Lihui Zhang; Jiangying Cao; Lei Zhang
作者单位1. School of Pharmacy Shandong Second Medical University Weifang Shandong China; 2. School of Stomatology Shandong Second Medical University Weifang Shandong China; 3. School of Pharmacy Shandong University of Traditional Chinese Medicine Jinan Shandong China
A Tale of Two Mechanisms: The p53 Modulator COTI‐2 Is a Zn Metallochaperone
作者İrem Şimşek; Farsheed Shahbazi‐Raz; Michael J. Krause; Azam Mohammadzadeh; Maryam Kosar; Peihan Xu; Samra Khan; Olena Tykhoniuk; Ashley DaDalt; Deya'a Almasri; Lara K. Watanabe; Kaitlyn Breault; John J. Hayward; Fraser S. Pick; Richard L. Ho; Jeremy M. Rawson; John F. Trant
作者单位1. Department of Chemistry and Biochemistry University of Windsor Windsor Ontario Canada; 2. Binary Star Research Services LaSalle Ontario Canada; 3. Department of Biomedical Sciences University of Windsor Windsor Ontario Canada; 4. Amaro Therapeutics New York New York USA; 5. WE‐Spark Research Institute Windsor Ontario Canada
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