医学
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20 篇有效样本 · 按发表日期由新到旧排列
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Synthesis of 1,3,5‐Triazine‐Indole Conjugates as Broad‐Spectrum Coronavirus Entry Inhibitors
作者Shazia Asghar; Leentje Persoons; Yanicka Smolders; Niels Willems; Dirk Daelemans; Steven De Jonghe; Najim A. Al‐Masoudi; Shahid Hameed
作者单位1. Department of Chemistry Quaid‐I‐Azam University Islamabad Pakistan; 2. Department of Microbiology, Immunology and Transplantation Rega Institute for Medical Research, Molecular Genetics and Therapeutics in Virology and Oncology Research Group, KU Leuven Leuven Belgium; 3. Department of Chemistry College of Science, University of Basrah Basrah Iraq
Tetramic Acid‐Derived Blue‐Emitting Fluorescent Probe for Selective Lipid Droplet Imaging in Live Cells and Zebrafish
作者Marija Grozdanić; Jelena Dinić; Miloš Jović; Ana Podolski‐Renić; Aleksandra Divac Rankov; Mila Ljujić; Milica Pešić; Igor M. Opsenica; Života Selaković
作者单位1. Institute for Biological Research “Siniša Stanković” – National Institute of the Republic of Serbia University of Belgrade Belgrade Serbia; 2. Innovative Centre of the Faculty of Chemistry University of Belgrade Belgrade Serbia; 3. Institute of Molecular Genetics and Genetic Engineering University of Belgrade Belgrade Serbia; 4. Department of Organic Chemistry University of Belgrade – Faculty of Chemistry Belgrade Serbia
Sugar Amino Acid Linkers for the Design of [ 18 F]SiFA‐PSMA Radioligands
作者Narendar R. Gade; Melinda Wuest; Justin J. Bailey; Atul Bhardwaj; Ralf Schirrmacher; Frank Wuest
作者单位1. Department of Oncology Cross Cancer Institute University of Alberta Edmonton Alberta Canada; 2. Department of Chemistry University of Alberta Edmonton Alberta Canada; 3. Cancer Research Institute of Northern Alberta Edmonton Alberta Canada
Deconstruction of Aspartic Protease Inhibitors Enables Fragment‐Based Discovery of Plasmepsin V Inhibitors
作者Marija Skvorcova; Laura Ruduša; Diana Zelencova‐Gopejenko; Aigars Jirgensons; Raitis Bobrovs
作者单位1. Latvian Institute of Organic Synthesis Riga Latvia; 2. Molport Inc. Riga Latvia
Novel Water‐Soluble, Heavy Atom‐Free Thioxanthene‐Fused Naphthalimide–Polyamine Phototheranostic Conjugates
作者Elisa Uliassi; Michele Rossi; Matteo Di Giosia; Amalia Conti; Matteo Calvaresi; Kerry J. Rhoden; Maria Laura Bolognesi
作者单位1. Department of Pharmacy and Biotechnology Alma Mater Studiorum ‐ University of Bologna Bologna Italy; 2. Department of Chemistry “Giacomo Ciamician” Alma Mater Studiorum ‐ University of Bologna Bologna Italy; 3. Preclinical & Translational Research in Oncology lab (PRO) IRCCS Azienda Ospedaliero ‐ Universitaria di Bologna Bologna Italy; 4. Medical Genetics Unit IRCCS Azienda Ospedaliero ‐ Universitaria di Bologna Bologna Italy; 5. Interdepartmental Center for Health Sciences & Technologies (HST), CIRI‐SDV Alma Mater Studiorum ‐ University of Bologna Bologna Italy; 6. Department of Medical and Surgical Sciences Alma Mater Studiorum ‐ University of Bologna Bologna Italy
Exploration of Nirmatrelvir Derivatives as Optimized SARS‐CoV‐2 Antivirals
作者Yugendar R. Alugubelli; Veerabhadra R. Vulupala; Kai S. Yang; Kaustav Khatua; Lauren R. Blankenship; Sathish Kumar; Demonta Coleman; Xuejiao Guo; Zhi Zachery Geng; Chia‐Chuan D. Cho; Banumathi Sankaran; Benjamin W. Neuman; Shiqing Xu; Wenshe Ray Liu
作者单位1. Texas A&M Drug Discovery Center Department of Chemistry College of Arts and Sciences Texas A&M University College Station Texas USA; 2. Department of Biology College of Arts and Sciences Texas A&M University College Station Texas USA; 3. Molecular Biophysics and Integrated Bioimaging Berkeley Center for Structural Biology Laurence Berkeley National Laboratory Berkeley California USA; 4. Texas A&M Global Health Research Complex Texas A&M University College Station Texas USA; 5. Department of Molecular Pathogenesis and Immunology College of Medicine Bryan Texas USA; 6. Department of Pharmaceutical Sciences Irma Lerma Rangel College of Pharmacy Texas A&M University College Station Texas USA; 7. Institute of Biosciences and Technology Department of Translational Medical Sciences School of Medicine Texas A&M University Houston Texas USA; 8. Department of Biochemistry and Biophysics College of Agriculture and Life Sciences Texas A&M University College Station Texas USA; 9. Department of Cell Biology and Genetics College of Medicine Texas A&M University College Station Texas USA
Design and Synthesis of Morroniside Derivatives Targeting H 2 O 2 ‐Induced Oxidative Stress: Antioxidant‐Triggered Neuroprotective Effect
作者Mingtao Wang; Haiyi Gao; Yuxiang Song; Baohong Sun; Yian Zhao; Peiliang Dong; Hua Han
作者单位1. College of Medicine Heilongjiang University of Chinese Medicine Harbin China; 2. Institute of Traditional Chinese Medicine Heilongjiang University of Chinese Medicine Harbin China
Rational Design of Multifunctional Tacrine Derivatives as Candidates for the Treatment of Alzheimer and Parkinson Diseases
作者Eugenia Dzib; Luis Felipe Hernández‐Ayala; Silvana Silva‐Aguirre; Annia Galano
作者单位1. Departamento de Química División de Ciencias Básicas e Ingeniería Universidad Autónoma Metropolitana, Unidad Iztapalapa Ciudad de México México; 2. Departamento de Física Aplicada Centro de Investigación y de Estudios Avanzados, Unidad Mérida Mérida Yucatán México
Hydroamination of Dehydroalanine With Deuterium Incorporation to Access Unnatural 2‐ and 4‐Pyridonyl α‐Amino Acids: Evaluation of Their Antibacterial, Antifungal, and Immunomodulatory Activities
作者Sowmya B. Udayakumar; Prakash Kumar; Karnati Sai Pranathi; Anjali Prajapati; Sunil Misra; Srinivasa Reddy Bonam; Kiranmai Nayani
作者单位1. Department of Organic Synthesis and Process Chemistry CSIR‐Indian Institute of Chemical Technology Hyderabad India; 2. Academy of Scientific and Innovative Research (AcSIR) Ghaziabad India; 3. Department of Applied Biology CSIR‐Indian Institute of Chemical Technology Hyderabad India; 4. Vaccine Immunology Laboratory Department of Applied Biology CSIR‐Indian Institute of Chemical Technology Hyderabad India
Structural and Functional Insights Into ( S )‐5′‐ C ‐Guanidinopropyl Uridine‐Modified Oligonucleotides With 2′‐ O ‐Methyl and 2′‐Fluoro Substitutions for RNAi Therapeutics
作者Sugahara Masaki; Elsayed M. Mahmoud; Shuichi Sakamoto; Yoshihito Ueno
作者单位1. United Graduate School of Agricultural Science Gifu University Gifu Japan; 2. Course of Applied Life Science Faculty of Applied Biological Sciences Gifu University Gifu Japan; 3. Department of Pharmaceutical Organic Chemistry Faculty of Pharmacy Zagazig University Zagazig Egypt; 4. Institute of Microbial Chemistry (BIKAKEN) Numazu Branch Microbial Chemistry Research Foundation Numazu Shizuoka Japan; 5. Department of Life Science and Chemistry The Graduate School of Natural Science and Technology Gifu University Gifu Japan; 6. Center for One Medicine Innovative Translational Research (COMIT) Tokai National Higher Education and Research System Gifu University Gifu Japan
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